產品屬性:
產品名稱 | NVS-CECR2-1 |
規格 | 1mg、5mg、10mg、25mg |
貨號 | EY-01Y12628 |
Cas No.: 1992047-61-6
別名: N/A
化學名: N/A
分子式: C27H37N5O2S

分子量: 495.7
溶解度: DMSO: 0.3 mg/mL
儲存條件: 4°C, protect from light
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述:
NVS-CECR2-1 is a potent inhibitor of CECR2 (cat eye syndrome chromosome region, candidate 2), a component of chromatin complexes that regulate gene expression controlling development. It binds CECR2 with high affinity (IC50 = 0.047 μM by Alpha screen, Kd = 0.80 μM by ITC). NVS-CECR2-1 demonstrates no crossreactivity in a panel of 48 bromodomains and has no major activity in kinase, protease, and receptor panels. It shows robust activity in cells by FRAP assay, due to its slow off-rate, and has no acute toxicity. See the Structural Genomics Consortium (SGC) website for more information.
特別提醒公司產品僅供科研使用